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  4. Activity of novel antibiotics against dual metallo-Beta-lactamase producing
    <i>Enterobacter hormaechei</i>
    clinical isolates
Details

Activity of novel antibiotics against dual metallo-Beta-lactamase producing <i>Enterobacter hormaechei</i> clinical isolates

Journal
JAC-Antimicrobial Resistance
ISSN
2632-1823
Date Issued
2026-01-07
Author(s)
Camila Solar
Facultad de Medicina Clínica Alemana Universidad del Desarrollo  
LORENA DIAZ BAYO
Facultad de Medicina Clínica Alemana Universidad del Desarrollo  
Katherine Soto
Facultad de Medicina Clínica Alemana Universidad del Desarrollo  
Jose R W Martínez
Facultad de Medicina Clínica Alemana Universidad del Desarrollo  
Nicolas Canales
Facultad de Medicina Clínica Alemana Universidad del Desarrollo  
Yehudit Bergman
Anne Peters
Facultad de Medicina Clínica Alemana Universidad del Desarrollo  
ARAOS BRALIC, RAFAEL IGNACIO  
Facultad de Medicina Clínica Alemana Universidad del Desarrollo  
Patricia García
Pranita D Tamma
MUNITA SEPULVEDA, JOSE MANUEL  
Facultad de Medicina Clínica Alemana Universidad del Desarrollo  
Type
journal-article
DOI
10.1093/jacamr/dlaf252
URL
https://hdl.handle.net/123456789/12161
Abstract
<jats:title>Abstract</jats:title>
<jats:sec>
<jats:title>Background</jats:title>
<jats:p>Metallo-β-lactamase (MBL)-producing carbapenemase-resistant Enterobacterales infections are associated with significant mortality. Several β-lactam/β-lactamase inhibitor combinations (BL/BLI) with promising activity against MBLs are in the pipeline.</jats:p>
</jats:sec>
<jats:sec>
<jats:title>Objective</jats:title>
<jats:p>To investigate the in vitro activity of upcoming BL/BLI agents against Enterobacter hormaechei clinical isolates co-producing NDM and VIM enzymes.</jats:p>
</jats:sec>
<jats:sec>
<jats:title>Methods</jats:title>
<jats:p>Eleven E. hormaechei isolates co-harbouring blaNDM-7 and blaVIM-1 were identified from 10 patients admitted to a tertiary hospital in Santiago, Chile, between July 2022 and July 2023. Reference broth microdilution (BMD) panels were developed to determine minimum inhibitory concentrations (MICs) to aztreonam/avibactam, cefepime/taniborbactam, cefepime/zidebactam, cefiderocol and cefiderocol/xeruborbactam. Cefiderocol population analysis profile–area under the curve (PAP–AUC) was performed in strains exhibiting cefiderocol susceptibility to assess for cefiderocol heteroresistance. Long-read sequencing, using the Oxford Nanopore Technologies platform, was conducted on all isolates to characterize the genomic background of blaNDM-7 and blaVIM-1.</jats:p>
</jats:sec>
<jats:sec>
<jats:title>Results</jats:title>
<jats:p>Among the 11 E. hormaechei isolates assemblies revealed blaNDM-7 and blaVIM-1 were located on separate plasmids. All isolates were susceptible to aztreonam/avibactam, cefepime/taniborbactam and cefepime/zidebactam. Cefiderocol susceptibility was variable; the addition of xeruborbactam restored susceptibility.</jats:p>
</jats:sec>
<jats:sec>
<jats:title>Conclusions</jats:title>
<jats:p>Our findings indicate that E. hormaechei clinical isolates co-producing NDM and VIM metallo-carbapenemases exhibited susceptibility to all tested novel BL/BLIs, including aztreonam/avibactam, cefepime/taniborbactam and cefepime/zidebactam. The combination of cefiderocol and xeruborbactam restored the activity of cefiderocol.</jats:p>
</jats:sec>
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